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Pharmacology & Toxicology
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Articles
Methods to accelerate PROTAC drug discovery
Open Access
Journal:
Biochemical Journal
Biochem J (2025) 482 (13): 921–937.
Published: 25 June 2025
Articles
Journal:
Biochemical Journal
Biochem J (2025) 482 (12): 839–857.
Published: 17 June 2025
Includes: Supplementary data
Articles
Insights into the cellular function and mechanism of action of quinone reductase 2 (NQO2)
Open Access
Journal:
Biochemical Journal
Biochem J (2025) 482 (06): 309–324.
Published: 11 March 2025
Articles
Opposing regulation of endoplasmic reticulum retention under stress by ERp44 and PDIA6
Available to PurchaseOlaya Yassin, Bellam Praveen, Odai Darawshi, Thomas LaFramboise, Miriam Shmuel, Shakti P. Pattanayak, Brian K. Law, Maria Hatzoglou, Boaz Tirosh
Journal:
Biochemical Journal
Biochem J (2024) 481 (24): 1921–1935.
Published: 09 December 2024
Includes: Supplementary data
Articles
Grace Q. Gong, Glenn R. Masson, Woo-Jeong Lee, James M. J. Dickson, Jackie D. Kendall, Manoj K. Rathinaswamy, Christina M. Buchanan, Martin Middleditch, Brady M. Owen, Julie A. Spicer, Gordon W. Rewcastle, William A. Denny, John E. Burke, Peter R. Shepherd, Roger L. Williams, Jack U. Flanagan
Journal:
Biochemical Journal
Biochem J (2024) 481 (23): 1787–1802.
Published: 28 November 2024
Includes: Supplementary data
Articles
Mitigating neuroinflammation in cognitive areas: exploring the impact of HMG-CoA reductase inhibitor
Available to PurchaseCarlos Henrique Rocha Catalão, Luis Henrique Angenendt da Costa, Jonathas Rodrigo dos Santos, Luciane Carla Alberici, Luiz Luciano Falconi-Sobrinho, Norberto Cysne Coimbra, Diogo Dominguini, Felipe Dal-Pizzol, Tatiana Barichello, Maria José Alves Rocha
Journal:
Biochemical Journal
Biochem J (2024) 481 (22): 1585–1602.
Published: 07 November 2024
Includes: Supplementary data
Articles
Jordana B. Freemantle, Dinesh Shah, Dylan M. Lynch, Alessio Ciulli, Harinder S. Hundal, D. Grahame Hardie
Journal:
Biochemical Journal
Biochem J (2024) 481 (18): 1203–1219.
Published: 12 September 2024
Includes: Supplementary data
Articles
Pregnane X receptor inhibits the transdifferentiation of hepatic stellate cells by down-regulating periostin expression
Available to PurchaseTakumi Sato, Ryota Shizu, Ryonosuke Baba, Akira Ooka, Takuomi Hosaka, Yuichiro Kanno, Kouichi Yoshinari
Journal:
Biochemical Journal
Biochem J (2024) 481 (18): 1173–1186.
Published: 06 September 2024
Includes: Supplementary data
Articles
Flaminia Mazzone, Astrid Hoeppner, Jens Reiners, Christoph G.W. Gertzen, Violetta Applegate, Mona A. Abdullaziz, Julia Gottstein, Daniel Degrandi, Martina Wesemann, Thomas Kurz, Sander H.J. Smits, Klaus Pfeffer
Journal:
Biochemical Journal
Biochem J (2024) 481 (16): 1075–1096.
Published: 21 August 2024
Includes: Supplementary data
Articles
Articles
Immunoregulatory signal networks and tumor immune evasion mechanisms: insights into therapeutic targets and agents in clinical development
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2022) 479 (20): 2219–2260.
Published: 28 October 2022
Articles
Immunothrombosis and the molecular control of tissue factor by pyroptosis: prospects for new anticoagulants
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2022) 479 (6): 731–750.
Published: 28 March 2022
Articles
Hiroko Otsuka, Hisashi Yokomizo, Shintaro Nakamura, Yoshihiro Izumi, Masatomo Takahashi, Sachiko Obara, Motonao Nakao, Yosuke Ikeda, Naoichi Sato, Ryuichi Sakamoto, Yasutaka Miyachi, Takashi Miyazawa, Takeshi Bamba, Yoshihiro Ogawa
Journal:
Biochemical Journal
Biochem J (2022) 479 (3): 425–444.
Published: 11 February 2022
Includes: Supplementary data
Articles
Pratiti Bhadra, Scott Dos Santos, Igor Gamayun, Tillman Pick, Clarissa Neumann, Joy Ogbechi, Belinda S. Hall, Richard Zimmermann, Volkhard Helms, Rachel E. Simmonds, Adolfo Cavalié
Journal:
Biochemical Journal
Biochem J (2021) 478 (22): 4005–4024.
Published: 23 November 2021
Includes: Supplementary data
Articles
Journal:
Biochemical Journal
Biochem J (2021) 478 (19): 3555–3573.
Published: 06 October 2021
Includes: Supplementary data
Articles
Conformational plasticity of the ULK3 kinase domain
Available to PurchaseSebastian Mathea, Eidarus Salah, Cynthia Tallant, Deep Chatterjee, Benedict-Tilman Berger, Rebecca Konietzny, Susanne Müller, Benedikt M. Kessler, Stefan Knapp
Journal:
Biochemical Journal
Biochem J (2021) 478 (14): 2811–2823.
Published: 23 July 2021
Includes: Supplementary data
Articles
The cAMP-phosphodiesterase 4 (PDE4) controls β-adrenoceptor- and CFTR-dependent saliva secretion in mice
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2021) 478 (10): 1891–1906.
Published: 24 May 2021
Includes: Supplementary data
Articles
Cancer cachexia: molecular mechanism and pharmacological management
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2021) 478 (9): 1663–1688.
Published: 10 May 2021
Articles
Rivastigmine attenuates the Alzheimer's disease related protein degradation and apoptotic neuronal death signalling
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2021) 478 (7): 1435–1451.
Published: 16 April 2021
Articles
Role of macrophage autophagy in atherosclerosis: modulation by bioactive compounds
Available to PurchaseMD Khurshidul Zahid, Hazera Binte Sufian, Mahua Choudhury, Masao Yamasaki, Ahmed Al-Harrasi, Naima Moustaid-Moussa, Shaikh Mizanoor Rahman
Journal:
Biochemical Journal
Biochem J (2021) 478 (7): 1359–1375.
Published: 16 April 2021
Articles
Sathish Sivaprakasam, Sabarish Ramachandran, Mohd Omar Faruk Sikder, Yangzom D. Bhutia, Mitchell W. Wachtel, Vadivel Ganapathy
Journal:
Biochemical Journal
Biochem J (2021) 478 (7): 1347–1358.
Published: 06 April 2021
Articles
Journal:
Biochemical Journal
Biochem J (2021) 478 (2): 389–406.
Published: 27 January 2021
Includes: Supplementary data
Articles
Heteromeric complex formation between human cytochrome P450 CYP1A1 and heme oxygenase-1
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2021) 478 (2): 377–388.
Published: 27 January 2021
Includes: Supplementary data
Articles
Modified organophosphorus fire retardant with low toxicity/high flame retardancy using the pharmacophore model associated with Mamdani fuzzy inference approach
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2020) 477 (23): 4655–4674.
Published: 11 December 2020
Includes: Supplementary data
Articles
Translesion synthesis of the major nitrogen mustard-induced DNA lesion by human DNA polymerase η
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2020) 477 (23): 4543–4558.
Published: 03 December 2020
Articles
Alexander Pflug, Marianne Schimpl, J. Willem M. Nissink, Ross C. Overman, Philip B. Rawlins, Caroline Truman, Elizabeth Underwood, Juli Warwicker, Jon Winter-Holt, William McCoull
Journal:
Biochemical Journal
Biochem J (2020) 477 (22): 4443–4452.
Published: 27 November 2020
Includes: Supplementary data
Articles
Kei Higuchi, Jonathan J. Kopel, Sathish Sivaprakasam, Valeria Jaramillo-Martinez, R. Bryan Sutton, Ina L. Urbatsch, Vadivel Ganapathy
Journal:
Biochemical Journal
Biochem J (2020) 477 (21): 4149–4165.
Published: 05 November 2020
Articles
Maurocalcin and its analog MCa E12A facilitate Ca 2+ mobilization in cardiomyocytes
Available to PurchaseStephan De Waard, Jérome Montnach, Charly Cortinovis, Olfa Chkir, Morteza Erfanian, Philippe Hulin, Nathalie Gaborit, Patricia Lemarchand, Pietro Mesirca, Isabelle Bidaud, Matteo E. Mangoni, Michel De Waard, Michel Ronjat
Journal:
Biochemical Journal
Biochem J (2020) 477 (20): 3985–3999.
Published: 29 October 2020
Includes: Supplementary data
Articles
Dopamine is an aryl hydrocarbon receptor agonist
Available to PurchaseHyejin Park, Un-ho Jin, Keshav Karki, Arul Jayaraman, Clint Allred, Sharon K. Michelhaugh, Sandeep Mittal, Robert S. Chapkin, Stephen Safe
Journal:
Biochemical Journal
Biochem J (2020) 477 (19): 3899–3910.
Published: 16 October 2020
Includes: Supplementary data
Articles
Journal:
Biochemical Journal
Biochem J (2020) 477 (18): 3583–3598.
Published: 28 September 2020
Includes: Supplementary data
Articles
Enantioseparation, in vitro testing, and structural characterization of triple-binding reactivators of organophosphate-inhibited cholinesterases
Available to PurchaseNikola Maraković, Anamarija Knežević, Igor Rončević, Xavier Brazzolotto, Zrinka Kovarik, Goran Šinko
Journal:
Biochemical Journal
Biochem J (2020) 477 (15): 2771–2790.
Published: 07 August 2020
Includes: Supplementary data
Articles
Impact of pesticide exposure on adipose tissue development and function
Available to PurchaseIn Collection
Adipose biology
Robert M. Gutgesell, Evangelia E. Tsakiridis, Shanza Jamshed, Gregory R. Steinberg, Alison C. Holloway
Journal:
Biochemical Journal
Biochem J (2020) 477 (14): 2639–2653.
Published: 29 July 2020
Articles
Cr(VI)-induced overactive mitophagy contributes to mitochondrial loss and cytotoxicity in L02 hepatocytes
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2020) 477 (14): 2607–2619.
Published: 24 July 2020
Articles
Articles
Interaction of the neutral amino acid transporter ASCT2 with basic amino acids
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2020) 477 (8): 1443–1457.
Published: 27 April 2020
Includes: Supplementary data
Articles
Sean Brennan, Hussein N. Rubaiy, Saba Imanzadeh, Ruth Reid, David Lodwick, Robert I. Norman, Richard D. Rainbow
Journal:
Biochemical Journal
Biochem J (2020) 477 (3): 671–689.
Published: 11 February 2020
Articles
Susanne Seemann, Mathias Ernst, Chiara Cimmaruta, Stephan Struckmann, Claudia Cozma, Dirk Koczan, Anne-Marie Knospe, Linda Rebecca Haake, Valentina Citro, Anja U. Bräuer, Giuseppina Andreotti, Maria Vittoria Cubellis, Georg Fuellen, Andreas Hermann, Anne-Katrin Giese, Arndt Rolfs, Jan Lukas
Journal:
Biochemical Journal
Biochem J (2020) 477 (2): 359–380.
Published: 30 January 2020
Includes: Supplementary data
Articles
Toward a systems approach to cytochrome P450 ensemble: interactions of CYP2E1 with other P450 species and their impact on CYP1A2
Available to PurchaseNadezhda Y. Davydova, Bikash Dangi, Marc A. Maldonado, Nikita E. Vavilov, Victor G. Zgoda, Dmitri R. Davydov
Journal:
Biochemical Journal
Biochem J (2019) 476 (23): 3661–3685.
Published: 12 December 2019
Includes: Supplementary data
Articles
Discovery of novel inhibitors of ribosome biogenesis by innovative high throughput screening strategies
Available to PurchaseCatherine E. Scull, Yinfeng Zhang, Nichole Tower, Lynn Rasmussen, Indira Padmalayam, Robert Hunter, Ling Zhai, Robert Bostwick, David A. Schneider
Journal:
Biochemical Journal
Biochem J (2019) 476 (15): 2209–2219.
Published: 09 August 2019
Includes: Supplementary data
Articles
Toxins for decoding interface selectivity in nicotinic acetylcholine receptors
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2019) 476 (10): 1515–1520.
Published: 28 May 2019
Articles
Glycolic acid attenuates UVB-induced aquaporin-3, matrix metalloproteinase-9 expression, and collagen degradation in keratinocytes and mouse skin
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2019) 476 (10): 1387–1400.
Published: 21 May 2019
Articles
Stephen Lynch, Chris S. Pridgeon, Carrie A. Duckworth, Parveen Sharma, B. Kevin Park, Chris E.P. Goldring
Journal:
Biochemical Journal
Biochem J (2019) 476 (7): 1149–1158.
Published: 15 April 2019
Articles
New insights into niclosamide action: autophagy activation in colorectal cancer
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2019) 476 (5): 779–781.
Published: 06 March 2019
Articles
Exosomal KLF3-AS1 from hMSCs promoted cartilage repair and chondrocyte proliferation in osteoarthritis
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2018) 475 (22): 3629–3638.
Published: 28 November 2018
Includes: Supplementary data
Articles
Role of ATP during the initiation of microvascularization: acceleration of an autocrine sensing mechanism facilitating chemotaxis by inorganic polyphosphate
Available to PurchaseWerner E.G. Müller, Maximilian Ackermann, Emad Tolba, Meik Neufurth, Ivan Ivetac, Maria Kokkinopoulou, Heinz C. Schröder, Xiaohong Wang
Journal:
Biochemical Journal
Biochem J (2018) 475 (20): 3255–3273.
Published: 31 October 2018
Articles
An Aβ42 variant that inhibits intra- and extracellular amyloid aggregation and enhances cell viability
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2018) 475 (19): 3087–3103.
Published: 10 October 2018
Includes: Supplementary data
Articles
In Collection
Editors' pick of research highlights published in the Biochemical Journal in 2018 & 2019
Dominic P. Byrne, Yong Li, Pawin Ngamlert, Krithika Ramakrishnan, Claire E. Eyers, Carrow Wells, David H. Drewry, William J. Zuercher, Neil G. Berry, David G. Fernig, Patrick A. Eyers
Journal:
Biochemical Journal
Biochem J (2018) 475 (15): 2435–2455.
Published: 14 August 2018
Includes: Supplementary data
Articles
Dominic P. Byrne, Yong Li, Krithika Ramakrishnan, Igor L. Barsukov, Edwin A. Yates, Claire E. Eyers, Dulcé Papy-Garcia, Sandrine Chantepie, Vijayakanth Pagadala, Jian Liu, Carrow Wells, David H. Drewry, William J. Zuercher, Neil G. Berry, David G. Fernig, Patrick A. Eyers
Journal:
Biochemical Journal
Biochem J (2018) 475 (15): 2417–2433.
Published: 14 August 2018
Includes: Supplementary data
Articles
The role of metabolism and tunneling nanotube-mediated intercellular mitochondria exchange in cancer drug resistance
Available to PurchaseIn Collection
Editors' pick of review article highlights published in the Biochemical Journal in 2018 & 2019
Journal:
Biochemical Journal
Biochem J (2018) 475 (14): 2305–2328.
Published: 31 July 2018
Articles
Stereochemistry as a determining factor for the effect of a cell-penetrating peptide on cellular viability and epithelial integrity
Available to Purchase
Journal:
Biochemical Journal
Biochem J (2018) 475 (10): 1773–1788.
Published: 24 May 2018
Includes: Supplementary data
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