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Recent advances in understanding GLP-1R (glucagon-like peptide-1 receptor) function

Biochem Soc Trans (2013) 41 (1): 172–179.
This article has been cited by the following articles in journals that are participating in CrossRef Cited-by Linking.
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  • An Xiang
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GSK-3 inhibition through GLP-1R allosteric activation mediates the neurogenesis promoting effect of P7C3 after cerebral ischemic/reperfusional injury in mice
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Discovery of a Novel Series of Orally Bioavailable and CNS Penetrant Glucagon-like Peptide-1 Receptor (GLP-1R) Noncompetitive Antagonists Based on a 1,3-Disubstituted-7-aryl-5,5-bis(trifluoromethyl)-5,8-dihydropyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione Core
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Liraglutide, a glucagon-like peptide-1 receptor agonist, facilitates osteogenic proliferation and differentiation in MC3T3-E1 cells through phosphoinositide 3-kinase (PI3K)/protein kinase B (AKT), extracellular signal-related kinase (ERK)1/2, and cAMP/protein kinase A (PKA) signaling pathways involving β-catenin
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Experimental Cell Research (2017) 360 (2): 281.
Genetically encoded photocross-linkers determine the biological binding site of exendin-4 peptide in the N-terminal domain of the intact human glucagon-like peptide-1 receptor (GLP-1R)
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Evidence for glucagon-like peptide-1 receptor signaling to activate ATP-sensitive potassium channels in pancreatic beta cells
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  • Seung Eun Song
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  • Dae-Kyu Song
Biochemical and Biophysical Research Communications (2016) 469 (2): 216.
A Hydrogen-Bonded Polar Network in the Core of the Glucagon-Like Peptide-1 Receptor Is a Fulcrum for Biased Agonism: Lessons from Class B Crystal Structures
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  • Christopher A. Reynolds
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  • Kevin J. Smith
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  • Tezz Quon
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  • Sebastian G.B. Furness
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Molecular Pharmacology (2016) 89 (3): 335.
Puerarin Protects Pancreatic β-Cells in Obese Diabetic Mice via Activation of GLP-1R Signaling
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Molecular Endocrinology (2016) 30 (3): 361.
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  • Jung-Mo Ahn
  • Jiayu Liao
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  • Caihong Zhou
  • Jiejie Deng
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  • Chuan He
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  • Patrick M. Sexton
  • Denise Wootten
  • Briony E. Forbes
  • Frank Grutzner
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  • Yuping Xu
  • Donghui Pan
  • Lizhen Wang
  • Runlin Yang
  • Chunjing Yu
  • Weixing Wan
  • Yiwei Wu
  • Min Yang
Biochemical and Biophysical Research Communications (2016) 471 (1): 47.
GPCR structure, function, drug discovery and crystallography: report from Academia-Industry International Conference (UK Royal Society) Chicheley Hall, 1–2 September 2014
  • Alexander Heifetz
  • Gebhard F. X. Schertler
  • Roland Seifert
  • Christopher G. Tate
  • Patrick M. Sexton
  • Vsevolod V. Gurevich
  • Daniel Fourmy
  • Vadim Cherezov
  • Fiona H. Marshall
  • R. Ian Storer
  • Isabel Moraes
  • Irina G. Tikhonova
  • Christofer S. Tautermann
  • Peter Hunt
  • Tom Ceska
  • Simon Hodgson
  • Mike J. Bodkin
  • Shweta Singh
  • Richard J. Law
  • Philip C. Biggin
Naunyn-Schmiedeberg's Archives of Pharmacology (2015) 388 (8): 883.
Cyclic alpha-conotoxin peptidomimetic chimeras as potent GLP-1R agonists
  • Joakim E. Swedberg
  • Christina I. Schroeder
  • Justin M. Mitchell
  • Thomas Durek
  • David P. Fairlie
  • David J. Edmonds
  • David A. Griffith
  • Roger B. Ruggeri
  • David R. Derksen
  • Paula M. Loria
  • Spiros Liras
  • David A. Price
  • David J. Craik
European Journal of Medicinal Chemistry (2015) 103: 175.
International Union of Basic and Clinical Pharmacology. XCIII. The Parathyroid Hormone Receptors—Family B G Protein–Coupled Receptors
  • Thomas J. Gardella
  • Jean-Pierre Vilardaga
Pharmacological Reviews (2015) 67 (2): 310.
Simultaneous determination of imigliptin and its three metabolites in human plasma and urine by liquid chromatography coupled to tandem mass spectrometry
  • Yang Liu
  • Dongyang Liu
  • Hongzhong Liu
  • Hanlin Song
  • Lin Song
  • Xueting Yao
  • Frank Wu
  • Chutian Shu
  • Xifeng Ma
  • Huimin Zhou
  • Ji Jiang
  • Pei Hu
Journal of Chromatography B (2015) 1002: 300.
Geniposide promotes beta-cell regeneration and survival through regulating β-catenin/TCF7L2 pathway
  • D D Yao
  • L Yang
  • Y Wang
  • C Liu
  • Y J Wei
  • X B Jia
  • W Yin
  • L Shu
Cell Death & Disease (2015) 6 (5): e1746.
New screening strategy and analysis for identification of allosteric modulators for glucagon-like peptide-1 receptor using GLP-1 (9-36) amide
  • Atsushi Nakane
  • Yusuke Gotoh
  • Junji Ichihara
  • Hidetaka Nagata
Analytical Biochemistry (2015) 491: 23.
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  • Print ISSN 0300-5127

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